(A) Lymphoma cell lines | ||||||
---|---|---|---|---|---|---|
EZH2 status | WSU-FSCLL | WILL1 | DOHH2 | SC1 | DB | SUDLH8 |
HKMT-I-005 | 3.405 | 5.599 | 3.257 | 3.711 | <1 | <1 |
GSK343 | 2.868 | 17.91 | 6.151 | 12.12. | <1 | 5.11 |
 | W.T. | W.T. | W.T. | W.T. | Mutant Y646N | W.T. |
(B) Breast cancer cell lines | ||||||
IC50 (μM) | MDA-MB-231 | MCF-7 | T-47D | BT-474 | SkBr3 | MCF10a |
HKMT-I-005 | 4.3 | 7.7 | 8.5 | 2.1 | 7.7 | >15 |